Ganirelix Powder Cas No.123246-29-7

Ganirelix Powder Cas No.123246-29-7

Khoom npe: Ganirelix Acetate Powder
Tau qhov twg los: Synthetic
Specification: Ntau dua lossis sib npaug li 99%
CAS Nr .: 123246-29-7
Molecular Formula: C₈₀H₁₁₃N₁₈O₁₃·2C₂H₄O₂ (nrog acetate)
Molecular Luj: ≈1690.4
Txoj Kev Xeem: HPLC
Cov khoom xyaw nquag: Ganirelix Acetate
Yam ntxwv: Dawb hmoov
Ntim: 1-100g; 1kg / aluminium ntawv ci hnab; 25kg / nruas
Cia txias: txias txias, tiv thaiv lub teeb, kaw, qhuav
Lub neej txee: 36 lub hlis

Kev Tshaj Tawm Txog Kev Siv: Cov khoom no yog tsim los siv rau kev lag luam lossis kev tshawb fawb tshawb fawb nkaus xwb.
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Khoom Description

 

Peb tshwj xeeb hauv kev tsim cov khoom lag luam siab-purity Ganirelix acetate active pharmaceutical ingredient (API), tsim nyob rau hauv nruj ua raws li kws tshuaj-qib cov qauv zoo. Tag nrho cov txheej txheem tsim khoom yog ua raws li cGMP kev taw qhia, kom ntseeg tau tias cov khoom tshwj xeeb homogeneity thiab batch-rau-batch sib xws. Peb Ganirelix acetate nthuav tawm cov tshuaj lom neeg thiab lom neeg ruaj khov, ua rau nws zoo tagnrho rau kev tsim kho.

Raws li tus neeg koom tes API ntseeg siab, peb tau cog lus los muab cov neeg siv khoom zoo, kev tswj hwm cov khoom lag luam los txhawb koj txoj kev loj hlob ruaj khov nyob rau hauv lub ntiaj teb kev pabcuam kev tsim cov cuab yeej cuab tam. Peb zoo siab tos txais koj cov lus nug thiab tos ntsoov rau kev sib koom tes.

Pharmacological Action

Ganirelix Acetate yog ib qho zoo heev Gonadotropin-Releasing Hormone (GnRH) antagonist. Nws lub luag haujlwm tseem ceeb yog ua kom sai thiab thim rov qab pituitary secretion ntawm Luteinizing Hormone (LH), yog li tiv thaiv kom tsis txhob muaj LH ntxov ntxov thaum lub sij hawm kho fertility. Cov nyhuv inhibitory meej no yog qhov tseem ceeb rau kev tswj hwm txoj kev loj hlob ntawm zes qe menyuam follicles.

Mechanism ntawm Action

Raws li ib qho hluavtaws decapeptide, Ganirelix Acetate ua haujlwm los ntawm kev sib tw thaiv GnRH receptors ntawm pituitary gonadotroph hlwb. Nws khi rau cov receptors nrog siab affinity, ncaj qha nyob ntawm qhov chaw receptor thiab tiv thaiv endogenous GnRH los ntawm kev khi. Txij li thaum nws tsis pib qhov pib "flare-up" cov nyhuv, nws tam sim ntawd suppresses tam sim ntawd suppresses lub secretion ntawm LH thiab Follicle-Stimulating Hormone (FSH), ua kom ceev hormonal tswj.

Product Efficiency

Cov txiaj ntsig tseem ceeb ntawm cov khoom no hauv kev kho mob daim ntawv thov yog kev tiv thaiv ntawm ovulation ntxov ntxov thaum tswj zes qe menyuam stimulation. Los ntawm kev tswj xyuas raws sij hawm, nws ua kom muaj ntau cov follicles tuaj yeem loj hlob tuaj, yog li ua rau oocyte retrieval tus nqi thiab tus naj npawb ntawm cov embryos zoo muaj rau kev hloov mus. Nws siv hauv Assisted Reproductive Technology pab txhim kho cov txheej txheem kho mob thiab txhim kho kev ua tiav tag nrho.

Khoom siv

Cov khoom no ua hauj lwm pab raws li ib tug Active Pharmaceutical Active Pharmaceutical Ingredient (API) tshwj xeeb yog siv nyob rau hauv formulation ntawm txhaj tshuaj npaj rau Assisted Reproductive Technology. Nws yog feem ntau qhia rau cov neeg mob infertile undergoing tswj zes qe menyuam stimulation, tswj nyob rau hauv lub nruab nrab-to-late theem ntawm stimulation raws tu qauv kom zoo tiv thaiv ib tug ntxov ntxov LH surge thiab xyuas kom meej kev vam meej ntawm lub qe retrieval txheej txheem. Nws cov haujlwm tshwj xeeb ua rau nws ua tus neeg sawv cev tseem ceeb hauv cov txheej txheem luv luv ntawm ovulation induction cycles.

 

Cim npe nrov: ganirelix hmoov cas no.123246-29-7, Tuam Tshoj ganirelix hmoov cas no.123246-29-7 manufacturers, lwm tus, Hoobkas

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