Acetyl Tetrapeptide-5 API Hmoov CAS 820959-17-9

Acetyl Tetrapeptide-5 API Hmoov CAS 820959-17-9

Acetyl Tetrapeptide-5 API|CAS Nr .: 820959-17-9 Periorbital Microcirculation Enhancer Acetyl Tetrapeptide-5 (kev lag luam hu ua Eyeseryl) yog ib qho tshwj xeeb hluavtaws tetrapeptide engineered los hais txog lub cev tsav tsheb ntawm periorbital edema thiab tsaus voj voog. Ntawm Xi'an Tihealth, ...
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High-Purity Acetyl Tetrapeptide-5 Powder CAS 820959-17-9

Acetyl Tetrapeptide-5 API|CAS Nr .: 820959-17-9 Periorbital Microcirculation Txhim Kho

Acetyl Tetrapeptide-5(kev lag luam hu ua Eyeseryl) yog ib qho tshwj xeeb hluavtaws tetrapeptide engineered los hais txog lub cev tsav tsheb ntawm periorbital edema thiab tsaus voj voog. Ntawm Xi'an Tihealth, peb muab qhov siab - specification API (C20H28N8O7) synthesized ntawm Khoom -Phase Peptide Synthesis (SPPS) nrog rau HPLC purity validated ntawm ntau dua los yog sib npaug rau 98.0%. Tsis zoo li cov pa ua kua dej, cov peptide no ua haujlwm raws li lub hom phiaj inhibitor ntawm vascular permeability thiab tus neeg saib xyuas antiglycation. Nws yog tsim tshwj xeeb rau siab -qhov muag kawg- kev saib xyuas uas muaj kev tswj xyuas meejhemodynamic fluxthiab collagen cross-kev sib txuas yuav tsum ua kom tiav qhov kev soj ntsuam xyuas kom txo tau qhov muag - lub ntim ntim.

⚠️ REGULATORY CEEB TOOM & Kev Tshawb Fawb Kev Tshawb Fawb

Kev Tshawb Fawb Tsuas Siv (RUO):Cov khoom no yog muab tshwj xeeb raws li ib tugraw khoom hmoovrau kev kuaj kev tshawb fawb thiab kev lag luam kws tshuaj. Nws yogTSIS TAUib qho khoom siv tiav tiav thiab nruj me ntsistxwv tsis pub siv ncaj qha rau tib neeg thov lossis nojnyob rau hauv nws daim ntawv tam sim no.

Risk Assumption:Tus neeg siv yuav luag txhua lub luag haujlwm rau kev tsim cov API no. Kev siv tsis raug, suav nrog kev sib cuag ntawm daim tawv nqaij ncaj qha yam tsis muaj chaw kho mob lossis cov khoom siv hluav taws xob tsis zoo, tuaj yeem ua rau khaus lossis ua tsis tiav.Xi'an Tihealth Biotechnology Co., Ltd. assumes tsis lavrau kev siv tsis tau tso cai lossis tsis yog - ua raws li kev tuav pov hwm.

Biochemical Mechanism thiab Vascular Permeability Control

Acetyl Tetrapeptide-5 attenuates qhov muag- lub hnab tsim los ntawm ob txoj kev ua haujlwm tsom rau cov kua tuav thiab cov ntaub so ntswg elasticity:

  • Anti-Edema Txoj Kev:Cov peptide inhibits qhov kev ua ntawm Angiotensin -Hloov Enzyme (ACE), yog li txo cov capillary permeability hauv cheeb tsam periorbital rhiab heev. Qhov no tiv thaiv lub extravasation ntawm cov kua rau hauv qhov chaw interstitial, txo qhov ntim ntawm lub qhov muag.
  • Kev tiv thaiv Antiglycation:Nws cuam tshuam nrog tus ntoo khaub lig- txuas ntawm collagen fibers los ntawm kev tiv thaiv cov txheej txheem glycation. Los ntawm kev tswj xyuas qhov yooj yim ntawm cov dermal matrix, nws ua kom cov tawv nqaij tseem muaj zog txaus los txhawb lub zos hemodynamic flux yam tsis muaj kev sib tsoo.
  • Kev kho dej kom zoo:Kev tshawb fawb soj ntsuam pom tau hais tias daim ntawv thov tsis tu ncua hauv lub tsheb xa khoom zoo txhawb nqa lymphatic kua, txo qhov pom ntawm cov voj voog tsaus ntuj los ntawm cov ntshav stasis thiab hyperpigmentation.

Formulation Parameters thiab Ionic Concentration Audit

Txhawm rau tswj hwm kev ua haujlwm lom neeg ntawm Acetyl Tetrapeptide-5, cov neeg tsim khoom yuav tsum ua raws li cov txheej txheem biophysical nruj thaum lub sijhawm tsim khoom:

CAS Nr 820959-17-9
HPLC Purity Ntau dua lossis sib npaug li 98.0%(Qhov tseeb ntawm RP-HPLC)
Molecular Luj 492.5 g / mol (qis dua 500 Da rau kev nkag mus zoo dua)
Ionic rhiab heev Siab; Yuav tsum nruj osmotic siab tswj
Residual acetic acid Tsawg dua los yog sib npaug li 8.0% (Tshem tawm cov qauv pH crashing)

Bench Note:Qhov no yog ibpH-sensitive additive. Qhov kawg bulk theem yuav tsum tau buffered ntawmpH 5.0 thiab 7.0. Lub zog ionic siab (salinity) hauv emulsion tuaj yeem ua rau peptide aggregation lossis poob ntawm kev tiv thaiv - edema potency. Kev sib xyaw ua ke ntawm qhov kub qis dua 35 degree.

Ntiaj teb no Kev Tshawb Fawb Kev Muag Khoom FAQ

Vim li cas Acetyl Tetrapeptide-5 rhiab heev rau ionic concentration ntawm cov mis?

Raws li me me -molecule peptide, nws qhov kev ruaj ntseg quaternary nyob ntawm qhov dielectric tas li ntawm cov kuab tshuaj. High electrolyte concentrations (ntsev) tuaj yeem cuam tshuam lub plhaub hydration ntawm peptide, ua rau muaj kev hloov pauv. Hauv qhov muag- cov qauv kev saib xyuas, qhov no feem ntau ua rau "stinging" hnov ​​​​qab rau qhov kawg- neeg siv lossis txo qis hauv vascular permeability efficiency.

Cov peptide no piv rau Caffeine li cas hauv kev tswj cov voj voog tsaus nti?

Caffeine feem ntau ua los ntawm vasoconstriction thiab stimulant ib ntus -raws li cov kua. Acetyl Tetrapeptide-5 muaj kev siv tshuaj muaj zog ntau dua los ntawm inhibiting glycation ntawm collagen thiab nquag txo qis vascular permeability. Nws hais txog qhovhauv pausntawm edema (kua kua) es tsis yog muab cov kua dej ib ntus.

Dab tsi yog qhov tseem ceeb ntawm "Acetic Acid" tswj rau qhov muag- cov qauv kev saib xyuas?

Residual acetic acid los ntawm theem synthesis yog ib qho kev khaus khaus. Peb Tsawg dua lossis sib npaug li 8.0% txwv yog qhov tseem ceeb rau qhov muag - daim ntawv thov hauv cheeb tsam kom ntseeg tau tias cov khoom kawg tsis ua rau lacrimation lossis periorbital erythema. Tsis tas li ntawd, nws tiv thaiv viscosity ntawm Carbomer-raws li qhov muag gels los ntawm ionic vau.

Puas yog Xi'an Tihealth muab cov ntaub ntawv ruaj ntseg rau kev tswj hwm thoob ntiaj teb?

Yog lawm. Peb muab tag nrho cov txheej txheem txheej txheem suav nrog HPLC chromatograms, MS cov ntaub ntawv, thiab luv luv - cov ntawv ceeb toom kev ruaj ntseg. Peb txhawb nqa peb cov koom tes thoob ntiaj teb nrog Batch Manufacturing Records (BMR) kom ua raws li cov kev soj ntsuam zoo uas yuav tsum tau muaj rau kev siv tshuaj thiab siab - kawg kev sau npe tshuaj pleev ib ce.

Xi'an Tihealth Biotechnology Ua raws li nqe lus:Raw khoom API rau kev lag luam R & D thiab kuaj siv xwb. Cov neeg siv xav tias txhua qhov kev pheej hmoo rau kev siv tshuaj kho mob tsis raug tso cai.

 
 
 
 

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